| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 1 |
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| Ligand | BDBM50244010 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_554820 (CHEMBL953973) |
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| Ki | 2396±n/a nM |
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| Citation |  Pagé, D; Balaux, E; Boisvert, L; Liu, Z; Milburn, C; Tremblay, M; Wei, Z; Woo, S; Luo, X; Cheng, YX; Yang, H; Srivastava, S; Zhou, F; Brown, W; Tomaszewski, M; Walpole, C; Hodzic, L; St-Onge, S; Godbout, C; Salois, D; Payza, K; Payza, K Novel benzimidazole derivatives as selective CB2 agonists. Bioorg Med Chem Lett18:3695-700 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 1 |
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| Name: | Cannabinoid receptor 1 |
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| Synonyms: | CANN6 | CANNABINOID CB1 | CB-R | CB1 | CNR | CNR1 | CNR1_HUMAN | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cannabinoid receptor 1 (brain) |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 52868.96 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P21554 |
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| Residue: | 472 |
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| Sequence: | MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQE
KMTAGDNPQLVPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIA
VLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVF
HRKDSRNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLM
WTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWK
AHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLL
AIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQ
PLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
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| BDBM50244010 |
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| n/a |
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| Name | BDBM50244010 |
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| Synonyms: | 2-(4-phenoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benzo[d]imidazole-5-carboxamide | CHEMBL510072 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H35N3O2 |
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| Mol. Mass. | 469.6178 |
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| SMILES | CCN(CC)C(=O)c1ccc2n(CCC(C)C)c(Cc3ccc(Oc4ccccc4)cc3)nc2c1 |
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| Structure | 
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