| Reaction Details |
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 | Report a problem with these data |
| Target | Monoglyceride lipase |
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| Ligand | BDBM50274151 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_537181 (CHEMBL992557) |
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| Ki | 58700±n/a nM |
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| Citation |  Magrioti, V; Naxakis, G; Hadjipavlou-Litina, D; Makriyannis, A; Kokotos, G A novel monoacylglycerol lipase inhibitor with analgesic and anti-inflammatory activity. Bioorg Med Chem Lett18:5424-7 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Monoglyceride lipase |
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| Name: | Monoglyceride lipase |
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| Synonyms: | MAGL | MGLL_RAT | Mgl2 | Mgll | Monoacylglycerol lipase | Monoglyceride lipase | Monoglyceride lipase (MGL) |
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| Type: | Enzyme |
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| Mol. Mass.: | 33505.38 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | Q8R431 |
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| Residue: | 303 |
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| Sequence: | MPEASSPRRTPQNVPYQDLPHLVNADGQYLFCRYWKPSGTPKALIFVSHGAGEHCGRYDE
LAQMLKRLDMLVFAHDHVGHGQSEGERMVVSDFQVFVRDLLQHVNTVQKDYPEVPVFLLG
HSMGGAISILAAAERPTHFSGMILISPLILANPESASTLKVLAAKLLNFVLPNISLGRID
SSVLSRNKSEVDLYNSDPLICHAGVKVCFGIQLLNAVSRVERAMPRLTLPFLLLQGSADR
LCDSKGAYLLMESSPSQDKTLKMYEGAYHVLHKELPEVTNSVLHEINTWVSHRIAVAGAR
CLP
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| BDBM50274151 |
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| n/a |
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| Name | BDBM50274151 |
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| Synonyms: | CHEMBL473249 | hexadecane-1,2-diamine dihydrochloride |
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| Type | Small organic molecule |
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| Emp. Form. | C16H36N2 |
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| Mol. Mass. | 256.4704 |
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| SMILES | CCCCCCCCCCCCCCC(N)CN |
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| Structure | 
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