| Reaction Details |
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 | Report a problem with these data |
| Target | Calcitonin gene-related peptide 1 |
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| Ligand | BDBM50246693 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_556932 (CHEMBL957387) |
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| IC50 | 8.9±n/a nM |
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| Citation |  Miranda, LP; Holder, JR; Shi, L; Bennett, B; Aral, J; Gegg, CV; Wright, M; Walker, K; Doellgast, G; Rogers, R; Li, H; Valladares, V; Salyers, K; Johnson, E; Wild, K Identification of potent, selective, and metabolically stable peptide antagonists to the calcitonin gene-related peptide (CGRP) receptor. J Med Chem51:7889-97 (2008) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Calcitonin gene-related peptide 1 |
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| Name: | Calcitonin gene-related peptide 1 |
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| Synonyms: | CALCA_RAT | CGRP | Calc | Calca | Calcitonin gene-related peptide 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 13950.43 |
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| Organism: | RAT |
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| Description: | CGRP 0 RAT::P01256 |
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| Residue: | 128 |
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| Sequence: | MGFLKFSPFLVVSILLLYQACGLQAVPLRSTLESSPGMAATLSEEEARLLLAALVQNYMQ
MKVRELEQEQEAEGSSVTAQKRSCNTATCVTHRLAGLLSRSGGVVKDNFVPTNVGSEAFG
RRRRDLQA
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| BDBM50246693 |
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| n/a |
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| Name | BDBM50246693 |
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| Synonyms: | Ac-WVTH[Cit]LAGLLS[Cit]SGGVVRKNFVPTDVGPFAF-NH2 | CHEMBL509329 |
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| Type | Small organic molecule |
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| Emp. Form. | C159H244N44O41 |
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| Mol. Mass. | 3427.9089 |
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| SMILES | n/a |
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| Structure | 
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