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TargetCalcitonin gene-related peptide 1
LigandBDBM50246695
Substrate/Competitorn/a
Meas. Tech.ChEMBL_556932 (CHEMBL957387)
IC50 20±n/a nM
Citation Miranda, LPHolder, JRShi, LBennett, BAral, JGegg, CVWright, MWalker, KDoellgast, GRogers, RLi, HValladares, VSalyers, KJohnson, EWild, K Identification of potent, selective, and metabolically stable peptide antagonists to the calcitonin gene-related peptide (CGRP) receptor. J Med Chem51:7889-97 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Calcitonin gene-related peptide 1
Name:Calcitonin gene-related peptide 1
Synonyms:CALCA_RAT | CGRP | Calc | Calca | Calcitonin gene-related peptide 1
Type:Enzyme Catalytic Domain
Mol. Mass.:13950.43
Organism:RAT
Description:CGRP 0 RAT::P01256
Residue:128
Sequence:
MGFLKFSPFLVVSILLLYQACGLQAVPLRSTLESSPGMAATLSEEEARLLLAALVQNYMQ
MKVRELEQEQEAEGSSVTAQKRSCNTATCVTHRLAGLLSRSGGVVKDNFVPTNVGSEAFG
RRRRDLQA
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BDBM50246695
n/a
NameBDBM50246695
Synonyms:Ac-WVTH[hArg]LAGLLS[hArg]SGGVVRKNFVPTDVGPFAF-NH2 | CHEMBL504769
TypeSmall organic molecule
Emp. Form.C161H250N46O39
Mol. Mass.3453.9925
SMILESn/a
Structure
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