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TargetCannabinoid receptor 2
LigandBDBM50277226
Substrate/Competitorn/a
Meas. Tech.ChEMBL_540512
Ki 85±n/a nM
Citation Goodman AJAjello CWWorm KLe Bourdonnec BSavolainen MAO'Hare HCassel JAStabley GJDehaven RNLabuda CJKoblish MLittle PJBrogdon BLSmith SADolle RE CB2 selective sulfamoyl benzamides: optimization of the amide functionality. Bioorg Med Chem Lett 19:309-13 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cannabinoid receptor 2
Name:Cannabinoid receptor 2
Synonyms:CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:G Protein-Coupled Receptor (GPCR)
Mol. Mass.:39690.94
Organism:Homo sapiens (Human)
Description:P34972
Residue:360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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BDBM50277226
n/a
NameBDBM50277226
Synonyms:4-(2-methyl-5-(5-neopentyl-1H-1,2,4-triazol-3-yl)phenylsulfonyl)morpholine | CHEMBL473697
TypeSmall organic molecule
Emp. Form.C18H26N4O3S
Mol. Mass.378.489
SMILESCc1ccc(cc1S(=O)(=O)N1CCOCC1)-c1nnc(CC(C)(C)C)[nH]1
Structure
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