| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50257851 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_567044 (CHEMBL1029952) |
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| Ki | 312±n/a nM |
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| Citation |  Zindell, R; Riether, D; Bosanac, T; Berry, A; Gemkow, MJ; Ebneth, A; Löbbe, S; Raymond, EL; Thome, D; Shih, DT; Thomson, D Morpholine containing CB2 selective agonists. Bioorg Med Chem Lett19:1604-9 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50257851 |
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| n/a |
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| Name | BDBM50257851 |
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| Synonyms: | (S)-4-((2',3'-dichlorobiphenyl-4-yl)methyl)-2-phenylmorpholine | CHEMBL494994 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H21Cl2NO |
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| Mol. Mass. | 398.325 |
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| SMILES | Clc1cccc(c1Cl)-c1ccc(CN2CCO[C@H](C2)c2ccccc2)cc1 |r| |
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| Structure | 
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