| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor M1 |
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| Ligand | BDBM50281908 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_139843 |
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| Kd | 679±n/a nM |
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| Citation |  Malaska, MJ; Fauq, AH; Kozikowski, AP; Aagaard, PJ; McKinney, M Simplified analogs of himbacine displaying potent binding affinity for muscarinic receptors Bioorg Med Chem Lett3:1247-1252 (1993) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Muscarinic acetylcholine receptor M1 |
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| Name: | Muscarinic acetylcholine receptor M1 |
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| Synonyms: | ACM1_HUMAN | CHRM1 | Cholinergic receptor, muscarinic 1 | Cholinergic, muscarinic M1 |
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| Type: | Protein |
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| Mol. Mass.: | 51442.54 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P11229 |
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| Residue: | 460 |
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| Sequence: | MNTSAPPAVSPNITVLAPGKGPWQVAFIGITTGLLSLATVTGNLLVLISFKVNTELKTVN
NYFLLSLACADLIIGTFSMNLYTTYLLMGHWALGTLACDLWLALDYVASNASVMNLLLIS
FDRYFSVTRPLSYRAKRTPRRAALMIGLAWLVSFVLWAPAILFWQYLVGERTVLAGQCYI
QFLSQPIITFGTAMAAFYLPVTVMCTLYWRIYRETENRARELAALQGSETPGKGGGSSSS
SERSQPGAEGSPETPPGRCCRCCRAPRLLQAYSWKEEEEEDEGSMESLTSSEGEEPGSEV
VIKMPMVDPEAQAPTKQPPRSSPNTVKRPTKKGRDRAGKGQKPRGKEQLAKRKTFSLVKE
KKAARTLSAILLAFILTWTPYNIMVLVSTFCKDCVPETLWELGYWLCYVNSTINPMCYAL
CNKAFRDTFRLLLLCRWDKRRWRKIPKRPGSVHRTPSRQC
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| BDBM50281908 |
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| n/a |
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| Name | BDBM50281908 |
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| Synonyms: | 2-((E)-2-Anthracen-9-yl-vinyl)-1-methyl-piperidine | CHEMBL22962 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H23N |
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| Mol. Mass. | 301.4247 |
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| SMILES | CN1CCCCC1\C=C\c1c2ccccc2cc2ccccc12 |
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| Structure | 
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