| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cholecystokinin receptor type A |
|---|
| Ligand | BDBM50283845 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_40039 |
|---|
| IC50 | 1.1±n/a nM |
|---|
| Citation |  Lowe, JA; Qian, W; Scott, PJ; McLean, S; Bryce, DK; Crawford, RT; Bordner, J 5,7-Diphenyl-3-ureidohexahydroazepin-2-ones as Cholecystokinin-B receptor ligands Bioorg Med Chem Lett4:2877-2882 (1994) Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cholecystokinin receptor type A |
|---|
| Name: | Cholecystokinin receptor type A |
|---|
| Synonyms: | CCK-A receptor | CCK-AR | CCK1-R | CCKAR | CCKAR_CAVPO | Cholecystokinin A receptor | Cholecystokinin receptor type A | Cholecystokinin-1 receptor |
|---|
| Type: | n/a |
|---|
| Mol. Mass.: | 48229.77 |
|---|
| Organism: | Cavia porcellus |
|---|
| Description: | n/a |
|---|
| Residue: | 430 |
|---|
| Sequence: | MDVVDSLFVNGSNITSACELGFENETLFCLDRPRPSKEWQPAVQILLYSLIFLLSVLGNT
LVITVLIRNKRMRTVTNIFLLSLAVSDLMLCLFCMPFNLIPSLLKDFIFGSAVCKTTTYF
MGTSVSVSTFNLVAISLERYGAICKPLQSRVWQTKSHALKVIAATWCLSFTIMTPYPIYS
NLVPFTKNNNQTGNMCRFLLPNDVMQQTWHTFLLLILFLIPGIVMMVAYGLISLELYQGI
KFDAIQKKSAKERKTSTGSSGPMEDSDGCYLQKSRHPRKLELRQLSPSSSGSNRINRIRS
SSSTANLMAKKRVIRMLIVIVVLFFLCWMPIFSANAWRAYDTVSAERHLSGTPISFILLL
SYTSSCVNPIIYCFMNKRFRLGFMATFPCCPNPGTPGVRGEMGEEEEGRTTGASLSRYSY
SHMSTSAPPP
|
|
|
|---|
| BDBM50283845 |
|---|
| n/a |
|---|
| Name | BDBM50283845 |
|---|
| Synonyms: | 2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-tolyl-ureido)-azepan-1-yl]-N-o-tolyl-acetamide | CHEMBL317615 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C36H38N4O3 |
|---|
| Mol. Mass. | 574.7119 |
|---|
| SMILES | Cc1cccc(NC(=O)N[C@@H]2C[C@@H](C[C@@H](N(CC(=O)Nc3ccccc3C)C2=O)c2ccccc2)c2ccccc2C)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
