| Reaction Details |
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 | Report a problem with these data |
| Target | Serotonin 1d (5-HT1d) receptor |
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| Ligand | BDBM50286672 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_1659 |
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| IC50 | 60±n/a nM |
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| Citation |  Perez M; Pauwels P; Palmier C; John GW; Valentin JP; Halazy S 5-O-Carboxymethyl piperazide derivatives of serotonin: a new class of potent and selective 5-HT1D receptor agonists Bioorg Med Chem Lett 5:663-666 (1995) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Serotonin 1d (5-HT1d) receptor |
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| Name: | Serotonin 1d (5-HT1d) receptor |
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| Synonyms: | 5-HT1D | 5-hydroxytryptamine receptor 1D | HTR1D |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 41780.38 |
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| Organism: | GUINEA PIG |
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| Description: | 5-HT1D HTR1D GUINEA PIG::Q60484 |
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| Residue: | 376 |
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| Sequence: | MSPPNQSEEGLPQEASNRSLNATETPGDWDPGLLQALKVSLVVVLSIITLATVLSNAFVL
TTILLTRKLHTPANYLIGSLATTDLLVSILVMPISIAYTTTRTWNFGQILCDIWVSSDIT
CCTASILHLCVIALDRYWAITDALEYSKRRTAGHAGAMIAAVWVISICISIPPLFWRQAQ
AQEEMSDCLVNTSQISYTIYSTCGAFYIPSVLLIILYSRIYRAARSRILNPPSLSGKRFT
TAHLITGSAGSSLCSLNPSLHEGHMHPGSPLFFNHVRIKLADSVLERKRISAARERKATK
TLGIILGAFIVCWLPFFVVSLVLPICRDSCWIHPALFDFFTWLGYLNSLINPIIYTVFNE
DFRQAFQKVVHFRKAS
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| BDBM50286672 |
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| n/a |
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| Name | BDBM50286672 |
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| Synonyms: | (S)-2-(2-{2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-acetylamino}-acetylamino)-3-(4-hydroxy-phenyl)-propionamide | CHEMBL159174 | GTI |
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| Type | Small organic molecule |
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| Emp. Form. | C23H27N5O5 |
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| Mol. Mass. | 453.491 |
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| SMILES | NCCc1c[nH]c2ccc(OCC(=O)NCC(=O)N[C@@H](Cc3ccc(O)cc3)C(N)=O)cc12 |
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| Structure | 
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