| Reaction Details |
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 | Report a problem with these data |
| Target | Chymotrypsin-like protease CTRL-1 |
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| Ligand | BDBM50288610 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_49606 (CHEMBL661257) |
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| IC50 | >1000±n/a nM |
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| Citation |  Iqbal, M; Chatterjee, S; Kauer, JC; Mallamo, JP; Messina, PA; Reiboldt, A; Siman, R Potent α-ketocarbonyl and boronic ester derived inhibitors of proteasome Bioorg Med Chem Lett6:287-290 (1996) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Chymotrypsin-like protease CTRL-1 |
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| Name: | Chymotrypsin-like protease CTRL-1 |
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| Synonyms: | CTRL | CTRL1 | CTRL_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 28008.18 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_49606 |
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| Residue: | 264 |
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| Sequence: | MLLLSLTLSLVLLGSSWGCGIPAIKPALSFSQRIVNGENAVLGSWPWQVSLQDSSGFHFC
GGSLISQSWVVTAAHCNVSPGRHFVVLGEYDRSSNAEPLQVLSVSRAITHPSWNSTTMNN
DVTLLKLASPAQYTTRISPVCLASSNEALTEGLTCVTTGWGRLSGVGNVTPAHLQQVALP
LVTVNQCRQYWGSSITDSMICAGGAGASSCQGDSGGPLVCQKGNTWVLIGIVSWGTKNCN
VRAPAVYTRVSKFSTWINQVIAYN
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| BDBM50288610 |
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| n/a |
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| Name | BDBM50288610 |
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| Synonyms: | Alpha-ketocarbonyl derivative | CHEMBL98937 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H50ClN7O5 |
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| Mol. Mass. | 612.204 |
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| SMILES | CC(C)CC(NC(=O)C(CCCN=C(N)N[N+]([O-])=O)NC(=O)C(CCCCCCCCC#N)C1CCCC1)C(=O)CCl |w:12.11| |
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| Structure | 
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