| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Casein kinase I isoform delta |
|---|
| Ligand | BDBM50299910 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_594445 (CHEMBL1041494) |
|---|
| IC50 | >1E4±n/a nM |
|---|
| Citation |  Okamoto, M; Takayama, K; Shimizu, T; Ishida, K; Takahashi, O; Furuya, T Identification of death-associated protein kinases inhibitors using structure-based virtual screening. J Med Chem52:7323-7 (2009) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Casein kinase I isoform delta |
|---|
| Name: | Casein kinase I isoform delta |
|---|
| Synonyms: | CKI-delta | CKId | CSNK1D | Casein kinase 1 delta (CK1δ) | Casein kinase I delta | Casein kinase I isoform alpha/delta | Casein kinase I isoform delta (CK1D) | HCKID | KC1D_HUMAN | casein kinases 1 delta (CK1 delta) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 47356.76 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P48730 |
|---|
| Residue: | 415 |
|---|
| Sequence: | MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQ
GGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIH
SKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYA
SINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVL
CKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRA
ADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEVAPPTPLTPTSHTANTSPRPV
SGMERERKVSMRLHRGAPVNISSSDLTGRQDTSRMSTSQIPGRVASSGLQSVVHR
|
|
|
|---|
| BDBM50299910 |
|---|
| n/a |
|---|
| Name | BDBM50299910 |
|---|
| Synonyms: | 4-(pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one | CHEMBL565286 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H12N2O2 |
|---|
| Mol. Mass. | 276.2894 |
|---|
| SMILES | O=C1OC(\C=C\c2ccccc2)=N/C/1=C\c1cccnc1 |c:12| |
|---|
| Structure | 
|
|---|
Search and Browse
