| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
|---|
| Ligand | BDBM50302306 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_596700 (CHEMBL1049670) |
|---|
| Ki | 1800±n/a nM |
|---|
| Citation |  Chu, GH; Saeui, CT; Worm, K; Weaver, DG; Goodman, AJ; Broadrup, RL; Cassel, JA; DeHaven, RN; LaBuda, CJ; Koblish, M; Brogdon, B; Smith, S; Le Bourdonnec, B; Dolle, RE Novel pyridine derivatives as potent and selective CB2 cannabinoid receptor agonists. Bioorg Med Chem Lett19:5931-5 (2009) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Cannabinoid receptor 2 |
|---|
| Name: | Cannabinoid receptor 2 |
|---|
| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 39690.94 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P34972 |
|---|
| Residue: | 360 |
|---|
| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
|
|
|
|---|
| BDBM50302306 |
|---|
| n/a |
|---|
| Name | BDBM50302306 |
|---|
| Synonyms: | 2,2-dimethyl-N-(5-methyl-6-(morpholinomethyl)pyridin-2-yl)butanamide | CHEMBL568146 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H27N3O2 |
|---|
| Mol. Mass. | 305.4152 |
|---|
| SMILES | CCC(C)(C)C(=O)Nc1ccc(C)c(CN2CCOCC2)n1 |
|---|
| Structure | 
|
|---|
Search and Browse
