| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 3 |
|---|
| Ligand | BDBM50304580 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_605121 (CHEMBL1073935) |
|---|
| IC50 | 752±n/a nM |
|---|
| Citation |  Fells, JI; Tsukahara, R; Liu, J; Tigyi, G; Parrill, AL Structure-based drug design identifies novel LPA3 antagonists. Bioorg Med Chem17:7457-64 (2009) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Lysophosphatidic acid receptor 3 |
|---|
| Name: | Lysophosphatidic acid receptor 3 |
|---|
| Synonyms: | EDG7 | LPA3 | LPAR3 | LPAR3_HUMAN | Lysophosphatidic acid receptor 1/3 | Lysophosphatidic acid receptor 3 (LPAR3) | Lysophosphatidic acid receptor Edg-7 |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 40149.72 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q9UBY5 |
|---|
| Residue: | 353 |
|---|
| Sequence: | MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNL
LVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDM
YGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
|
|
|
|---|
| BDBM50304580 |
|---|
| n/a |
|---|
| Name | BDBM50304580 |
|---|
| Synonyms: | 2-(3-(4-nitrophenoxy)phenyl)-1,3-dioxoisoindoline-5-carboxylic acid | CHEMBL604677 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H12N2O7 |
|---|
| Mol. Mass. | 404.3292 |
|---|
| SMILES | OC(=O)c1ccc2C(=O)N(C(=O)c2c1)c1cccc(Oc2ccc(cc2)[N+]([O-])=O)c1 |
|---|
| Structure | 
|
|---|
Search and Browse
