| Reaction Details |
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 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 5 |
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| Ligand | BDBM50304580 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_605123 (CHEMBL1064666) |
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| IC50 | 463±n/a nM |
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| Citation |  Fells, JI; Tsukahara, R; Liu, J; Tigyi, G; Parrill, AL Structure-based drug design identifies novel LPA3 antagonists. Bioorg Med Chem17:7457-64 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Lysophosphatidic acid receptor 5 |
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| Name: | Lysophosphatidic acid receptor 5 |
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| Synonyms: | GPR92 | GPR93 | LPAR5 | LPAR5_HUMAN | Lysophosphatidic acid receptor 5 | Lysophosphatidic acid receptor 5 (LPA5) |
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| Type: | Enzyme |
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| Mol. Mass.: | 41372.36 |
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| Organism: | Homo sapiens (Human) |
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| Description: | Q9H1C0 |
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| Residue: | 372 |
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| Sequence: | MLANSSSTNSSVLPCPDYRPTHRLHLVVYSLVLAAGLPLNALALWVFLRALRVHSVVSVY
MCNLAASDLLFTLSLPVRLSYYALHHWPFPDLLCQTTGAIFQMNMYGSCIFLMLINVDRY
AAIVHPLRLRHLRRPRVARLLCLGVWALILVFAVPAARVHRPSRCRYRDLEVRLCFESFS
DELWKGRLLPLVLLAEALGFLLPLAAVVYSSGRVFWTLARPDATQSQRRRKTVRLLLANL
VIFLLCFVPYNSTLAVYGLLRSKLVAASVPARDRVRGVLMVMVLLAGANCVLDPLVYYFS
AEGFRNTLRGLGTPHRARTSATNGTRAALAQSERSAVTTDATRPDAASQGLLRPSDSHSL
SSFTQCPQDSAL
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| BDBM50304580 |
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| n/a |
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| Name | BDBM50304580 |
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| Synonyms: | 2-(3-(4-nitrophenoxy)phenyl)-1,3-dioxoisoindoline-5-carboxylic acid | CHEMBL604677 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H12N2O7 |
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| Mol. Mass. | 404.3292 |
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| SMILES | OC(=O)c1ccc2C(=O)N(C(=O)c2c1)c1cccc(Oc2ccc(cc2)[N+]([O-])=O)c1 |
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| Structure | 
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