| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Lysophosphatidic acid receptor 3 |
|---|
| Ligand | BDBM50271701 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_605121 (CHEMBL1073935) |
|---|
| IC50 | 30±n/a nM |
|---|
| Citation |  Fells, JI; Tsukahara, R; Liu, J; Tigyi, G; Parrill, AL Structure-based drug design identifies novel LPA3 antagonists. Bioorg Med Chem17:7457-64 (2009) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Lysophosphatidic acid receptor 3 |
|---|
| Name: | Lysophosphatidic acid receptor 3 |
|---|
| Synonyms: | EDG7 | LPA3 | LPAR3 | LPAR3_HUMAN | Lysophosphatidic acid receptor 1/3 | Lysophosphatidic acid receptor 3 (LPAR3) | Lysophosphatidic acid receptor Edg-7 |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 40149.72 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q9UBY5 |
|---|
| Residue: | 353 |
|---|
| Sequence: | MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNL
LVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDM
YGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
|
|
|
|---|
| BDBM50271701 |
|---|
| n/a |
|---|
| Name | BDBM50271701 |
|---|
| Synonyms: | 2,6-bis(3-carboxyacrylamido)benzoic acid | 4,4'-(2-carboxy-1,3-phenylene)bis(azanediyl)bis(4-oxobut-2-enoic acid) | CHEMBL485119 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C15H12N2O8 |
|---|
| Mol. Mass. | 348.2644 |
|---|
| SMILES | OC(=O)\C=C\C(=O)Nc1cccc(NC(=O)\C=C\C(O)=O)c1C(O)=O |
|---|
| Structure | 
|
|---|
Search and Browse
