| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Urotensin-2 receptor |
|---|
| Ligand | BDBM50320467 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_636751 (CHEMBL1167040) |
|---|
| Ki | 610±n/a nM |
|---|
| Citation |  Maryanoff, BE; Kinney, WA Urotensin-II receptor modulators as potential drugs. J Med Chem53:2695-708 (2010) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Urotensin-2 receptor |
|---|
| Name: | Urotensin-2 receptor |
|---|
| Synonyms: | G-protein coupled receptor 14 | G-protein coupled sensory epithelial neuropeptide-like receptor | Gpr14 | Senr | UR-II-R | UR2R_RAT | Urotensin-II | Uts2r |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 42725.34 |
|---|
| Organism: | RAT |
|---|
| Description: | Urotensin-II UTS2R RAT::P49684 |
|---|
| Residue: | 386 |
|---|
| Sequence: | MALSLESTTSFHMLTVSGSTVTELPGDSNVSLNSSWSGPTDPSSLKDLVATGVIGAVLSA
MGVVGMVGNVYTLVVMCRFLRASASMYVYVVNLALADLLYLLSIPFIIATYVTKDWHFGD
VGCRVLFSLDFLTMHASIFTLTIMSSERYAAVLRPLDTVQRSKGYRKLLVLGTWLLALLL
TLPMMLAIQLVRRGSKSLCLPAWGPRAHRTYLTLLFGTSIVGPGLVIGLLYVRLARAYWL
SQQASFKQTRRLPNPRVLYLILGIVLLFWACFLPFWLWQLLAQYHEAMPLTPETARIVNY
LTTCLTYGNSCINPFLYTLLTKNYREYLRGRQRSLGSSCHSPGSPGSFLPSRVHLQQDSG
RSLSSSSQQATETLMLSPVPRNGALL
|
|
|
|---|
| BDBM50320467 |
|---|
| n/a |
|---|
| Name | BDBM50320467 |
|---|
| Synonyms: | Ac-[CFwKYC]-NH2 | CHEMBL1163477 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C43H53N9O8S2 |
|---|
| Mol. Mass. | 888.066 |
|---|
| SMILES | CC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC1=O)C(N)=O |r| |
|---|
| Structure | 
|
|---|
Search and Browse
