| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50325533 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_652218 (CHEMBL1228491) |
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| Ki | 5.85±n/a nM |
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| Citation |  Fujii, H; Ida, Y; Hanamura, S; Osa, Y; Nemoto, T; Nakajima, M; Hasebe, K; Nakao, K; Mochizuki, H; Nagase, H Synthesis of pyrrolomorphinan derivatives as kappa opioid agonists. Bioorg Med Chem Lett20:5035-8 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50325533 |
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| n/a |
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| Name | BDBM50325533 |
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| Synonyms: | CHEMBL1223890 |
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| Type | Small organic molecule |
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| Emp. Form. | C28H34N2O3 |
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| Mol. Mass. | 446.5812 |
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| SMILES | CCC\C=C\c1cc2C[C@@]3(O)[C@H]4Cc5ccc(O)c6O[C@@H](c2n1C)[C@]3(CCN4CC1CC1)c56 |r| |
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| Structure | 
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