| Reaction Details |
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 | Report a problem with these data |
| Target | Cannabinoid receptor 2 |
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| Ligand | BDBM50332256 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_685961 (CHEMBL1292717) |
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| Ki | 2040±n/a nM |
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| Citation |  Osman, NA; Mahmoud, AH; Allarà, M; Niess, R; Abouzid, KA; Di Marzo, V; Abadi, AH Synthesis, binding studies and molecular modeling of novel cannabinoid receptor ligands. Bioorg Med Chem18:8463-77 (2010) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Cannabinoid receptor 2 |
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| Name: | Cannabinoid receptor 2 |
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| Synonyms: | CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 39690.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P34972 |
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| Residue: | 360 |
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| Sequence: | MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILS
SHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTAS
VGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCS
ELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLD
VRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYA
LRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
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| BDBM50332256 |
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| n/a |
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| Name | BDBM50332256 |
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| Synonyms: | (E)-7-Naphthalen-2-yl-5-oxohept-6-enoic acid cyclopropylamide | CHEMBL1288209 |
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| Type | Small organic molecule |
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| Emp. Form. | C20H21NO2 |
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| Mol. Mass. | 307.3862 |
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| SMILES | O=C(CCCC(=O)C=Cc1ccc2ccccc2c1)NC1CC1 |w:8.8| |
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| Structure | 
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