| Reaction Details |
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 | Report a problem with these data |
| Target | Phospholipase A2 group V |
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| Ligand | BDBM50333788 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_700980 (CHEMBL1648640) |
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| IC50 | 2600±n/a nM |
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| Citation |  Mouchlis, VD; Magrioti, V; Barbayianni, E; Cermak, N; Oslund, RC; Mavromoustakos, TM; Gelb, MH; Kokotos, G Inhibition of secreted phospholipases A2 by 2-oxoamides based ona-amino acids: Synthesis, in vitro evaluation and molecular docking calculations. Bioorg Med Chem19:735-43 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Phospholipase A2 group V |
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| Name: | Phospholipase A2 group V |
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| Synonyms: | PA2G5_MOUSE | Pla2g5 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 15864.30 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_700980 |
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| Residue: | 137 |
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| Sequence: | MKGLLTLAWFLACSVPAVPGGLLELKSMIEKVTGKNAFKNYGFYGCYCGWGGRGTPKDGT
DWCCQMHDRCYGQLEEKDCAIRTQSYDYRYTNGLVICEHDSFCPMRLCACDRKLVYCLRR
NLWTYNPLYQYYPNFLC
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| BDBM50333788 |
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| n/a |
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| Name | BDBM50333788 |
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| Synonyms: | (S)-4-Methyl-2-(2-oxohexadecanamido)pentanoic acid | CHEMBL1644549 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H41NO4 |
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| Mol. Mass. | 383.5652 |
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| SMILES | CCCCCCCCCCCCCCC(=O)C(=O)N[C@@H](CC(C)C)C(O)=O |r| |
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| Structure | 
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