| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50336677 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_722917 (CHEMBL1674428) |
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| Ki | 0.182±n/a nM |
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| Citation |  Nemoto, T; Yamamoto, N; Watanabe, A; Fujii, H; Hasebe, K; Nakajima, M; Mochizuki, H; Nagase, H Synthesis of 6,14-epoxymorphinan derivatives and their pharmacologies. Bioorg Med Chem19:1205-21 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50336677 |
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| n/a |
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| Name | BDBM50336677 |
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| Synonyms: | CHEMBL1672484 | N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3-hydroxymorphinan-6alpha-yl)methyl]-3-phenylpropionamide |
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| Type | Small organic molecule |
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| Emp. Form. | C30H36N2O3 |
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| Mol. Mass. | 472.6184 |
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| SMILES | Oc1ccc2C[C@H]3N(CC4CC4)CC[C@@]4(C[C@]5(CNC(=O)CCc6ccccc6)CC[C@@]34O5)c2c1 |r,THB:8:7:31:33.4.5| |
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| Structure | 
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