| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin E2 receptor EP2 subtype |
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| Ligand | BDBM50351477 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_764671 (CHEMBL1821223) |
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| Ki | 3500±n/a nM |
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| Citation |  Iwahashi, M; Takahashi, E; Tanaka, M; Matsunaga, Y; Okada, Y; Matsumoto, R; Nambu, F; Nakai, H; Toda, M Design and synthesis of new prostaglandin D2 receptor antagonists. Bioorg Med Chem19:5361-71 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin E2 receptor EP2 subtype |
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| Name: | Prostaglandin E2 receptor EP2 subtype |
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| Synonyms: | PE2R2_MOUSE | PGE receptor, EP2 subtype | Prostaglandin E2 | Prostaglandin E2 receptor EP2 subtype | Prostanoid EP2 receptor | Ptger2 | Ptgerep2 |
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| Type: | G-protein coupled receptor |
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| Mol. Mass.: | 40495.26 |
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| Organism: | Mus musculus (Mouse) |
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| Description: | n/a |
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| Residue: | 362 |
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| Sequence: | MDNFLNDSKLMEDCKSRQWLLSGESPAISSVMFSAGVLGNLIALALLARRWRGDTGCSAG
SRTSISLFHVLVTELVLTDLLGTCLISPVVLASYSRNQTLVALAPESHACTYFAFTMTFF
SLATMLMLFAMALERYLSIGYPYFYRRHLSRRGGLAVLPVIYGASLLFCSLPLLNYGEYV
QYCPGTWCFIRHGRTAYLQLYATMLLLLIVAVLACNISVILNLIRMHRRSRRSRCGLSGS
SLRGPGSRRRGERTSMAEETDHLILLAIMTITFAICSLPFTIFAYMDETSSLKEKWDLRA
LRFLSVNSIIDPWVFAILRPPVLRLMRSVLCCRTSLRTQEAQQTSCSTQSSASKQTDLCG
QL
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| BDBM50351477 |
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| n/a |
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| Name | BDBM50351477 |
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| Synonyms: | CHEMBL1819605 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H24N2O5 |
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| Mol. Mass. | 432.4685 |
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| SMILES | CN1C[C@@H](COc2ccc(NC(=O)c3cccc(CC(O)=O)c3)cc2)Oc2ccccc12 |r| |
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| Structure | 
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