| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin F2-alpha receptor |
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| Ligand | BDBM50152515 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_764677 (CHEMBL1821229) |
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| Ki | 3100±n/a nM |
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| Citation |  Iwahashi, M; Takahashi, E; Tanaka, M; Matsunaga, Y; Okada, Y; Matsumoto, R; Nambu, F; Nakai, H; Toda, M Design and synthesis of new prostaglandin D2 receptor antagonists. Bioorg Med Chem19:5361-71 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin F2-alpha receptor |
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| Name: | Prostaglandin F2-alpha receptor |
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| Synonyms: | PF2R_MOUSE | ProstaglandinF2Alpha | Ptgfr |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40714.02 |
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| Organism: | MOUSE |
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| Description: | ProstaglandinF2Alpha PTGFR MOUSE::P43117 |
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| Residue: | 366 |
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| Sequence: | MSMNSSKQPVSPAAGLIANTTCQTENRLSVFFSIIFMTVGILSNSLAIAILMKAYQRFRQ
KSKASFLLLASGLVITDFFGHLINGGIAVFVYASDKDWIRFDQSNILCSIFGISMVFSGL
CPLFLGSAMAIERCIGVTNPIFHSTKITSKHVKMILSGVCMFAVFVAVLPILGHRDYQIQ
ASRTWCFYNTEHIEDWEDRFYLLFFSFLGLLALGVSFSCNAVTGVTLLRVKFRSQQHRQG
RSHHLEMIIQLLAIMCVSCVCWSPFLVTMANIAINGNNSPVTCETTLFALRMATWNQILD
PWVYILLRKAVLRNLYKLASRCCGVNIISLHIWELSSIKNSLKVAAISESPAAEKESQQA
SSEAGL
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| BDBM50152515 |
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| n/a |
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| Name | BDBM50152515 |
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| Synonyms: | CHEMBL364841 | {2-Methyl-1-[4-(4-methyl-3,4-dihydro-2H-benzo[1,4]oxazin-2-ylmethoxy)-benzoyl]-1H-indol-4-yl}-acetic acid |
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| Type | Small organic molecule |
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| Emp. Form. | C28H26N2O5 |
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| Mol. Mass. | 470.5164 |
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| SMILES | CN1C[C@@H](COc2ccc(cc2)C(=O)n2c(C)cc3c(CC(O)=O)cccc23)Oc2ccccc12 |
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| Structure | 
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