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TargetTranscriptional activator protein LasR
LigandBDBM50350703
Substrate/Competitorn/a
Meas. Tech.ChEMBL_765284 (CHEMBL1827923)
EC50 7±n/a nM
Citation Lowery, CASalzameda, NTSawada, DKaufmann, GFJanda, KD Medicinal chemistry as a conduit for the modulation of quorum sensing. J Med Chem53:7467-89 (2010) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Transcriptional activator protein LasR
Name:Transcriptional activator protein LasR
Synonyms:LASR_PSEAE | lasR
Type:PROTEIN
Mol. Mass.:26618.24
Organism:Pseudomonas aeruginosa
Description:ChEMBL_1475312
Residue:239
Sequence:
MALVDGFLELERSSGKLEWSAILQKMASDLGFSKILFGLLPKDSQDYENAFIVGNYPAAW
REHYDRAGYARVDPTVSHCTQSVLPIFWEPSIYQTRKQHEFFEEASAAGLVYGLTMPLHG
ARGELGALSLSVEAENRAEANRFMESVLPTLWMLKDYALQSGAGLAFEHPVSKPVVLTSR
EKEVLQWCAIGKTSWEISVICNCSEANVNFHMGNIRRKFGVTSRRVAAIMAVNLGLITL
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BDBM50350703
n/a
NameBDBM50350703
Synonyms:CHEMBL1814828
TypeSmall organic molecule
Emp. Form.C16H27NO3S
Mol. Mass.313.455
SMILESCCCCCCCCCC(=O)CC(=O)N[C@H]1CCSC1=O |r|
Structure
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