| Reaction Details |
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 | Report a problem with these data |
| Target | UDP-glucuronosyltransferase 2B7 |
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| Ligand | BDBM50003616 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_774127 (CHEMBL1908132) |
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| Ki | 1600000±n/a nM |
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| Citation |  Kiang, TK; Ensom, MH; Chang, TK UDP-glucuronosyltransferases and clinical drug-drug interactions. Pharmacol Ther106:97-132 (2005) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| UDP-glucuronosyltransferase 2B7 |
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| Name: | UDP-glucuronosyltransferase 2B7 |
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| Synonyms: | 2.4.1.17 | 3,4-catechol estrogen-specific UDPGT | UD2B7_HUMAN | UDP-glucuronosyltransferase 2B7 | UDP-glucuronosyltransferase 2B9 | UDPGT 2B7 | UDPGT 2B9 | UDPGTh-2 | UGT2B7 | UGTB2B9 | Uridine-5'-diphosphoglucuronosyltransferase 2B7 |
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| Type: | Enzyme |
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| Mol. Mass.: | 60705.98 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P16662 |
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| Residue: | 529 |
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| Sequence: | MSVKWTSVILLIQLSFCFSSGNCGKVLVWAAEYSHWMNIKTILDELIQRGHEVTVLASSA
SILFDPNNSSALKIEIYPTSLTKTELENFIMQQIKRWSDLPKDTFWLYFSQVQEIMSIFG
DITRKFCKDVVSNKKFMKKVQESRFDVIFADAIFPCSELLAELFNIPFVYSLSFSPGYTF
EKHSGGFIFPPSYVPVVMSELTDQMTFMERVKNMIYVLYFDFWFEIFDMKKWDQFYSEVL
GRPTTLSETMGKADVWLIRNSWNFQFPYPLLPNVDFVGGLHCKPAKPLPKEMEDFVQSSG
ENGVVVFSLGSMVSNMTEERANVIASALAQIPQKVLWRFDGNKPDTLGLNTRLYKWIPQN
DLLGHPKTRAFITHGGANGIYEAIYHGIPMVGIPLFADQPDNIAHMKARGAAVRVDFNTM
SSTDLLNALKRVINDPSYKENVMKLSRIQHDQPVKPLDRAVFWIEFVMRHKGAKHLRVAA
HDLTWFQYHSLDVIGFLLVCVATVIFIVTKCCLFCFWKFARKAKKGKND
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| BDBM50003616 |
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| n/a |
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| Name | BDBM50003616 |
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| Synonyms: | 2-n-propyl-n-valeric acid | CHEMBL109 | DPA | Di-n-propylessigsaeure | VALPROIC ACID | Valproinsaeure | dipropylacetic acid | n-DPA |
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| Type | Small organic molecule |
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| Emp. Form. | C8H16O2 |
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| Mol. Mass. | 144.2114 |
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| SMILES | CCCC(CCC)C(O)=O |
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| Structure | 
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