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TargetSerine/threonine-protein kinase 38-like
LigandBDBM60589
Substrate/Competitorn/a
Meas. Tech.ChEMBL_774572 (CHEMBL1908789)
Kd>10000±n/a nM
Citation Davis, MIHunt, JPHerrgard, SCiceri, PWodicka, LMPallares, GHocker, MTreiber, DKZarrinkar, PP Comprehensive analysis of kinase inhibitor selectivity. Nat Biotechnol29:1046-51 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Serine/threonine-protein kinase 38-like
Name:Serine/threonine-protein kinase 38-like
Synonyms:KIAA0965 | NDR2 | ST38L_HUMAN | STK38L
Type:PROTEIN
Mol. Mass.:54004.24
Organism:Homo sapiens (Human)
Description:ChEMBL_587191
Residue:464
Sequence:
MAMTAGTTTTFPMSNHTRERVTVAKLTLENFYSNLILQHEERETRQKKLEVAMEEEGLAD
EEKKLRRSQHARKETEFLRLKRTRLGLDDFESLKVIGRGAFGEVRLVQKKDTGHIYAMKI
LRKSDMLEKEQVAHIRAERDILVEADGAWVVKMFYSFQDKRNLYLIMEFLPGGDMMTLLM
KKDTLTEEETQFYISETVLAIDAIHQLGFIHRDIKPDNLLLDAKGHVKLSDFGLCTGLKK
AHRTEFYRNLTHNPPSDFSFQNMNSKRKAETWKKNRRQLAYSTVGTPDYIAPEVFMQTGY
NKLCDWWSLGVIMYEMLIGYPPFCSETPQETYRKVMNWKETLVFPPEVPISEKAKDLILR
FCIDSENRIGNSGVEEIKGHPFFEGVDWEHIRERPAAIPIEIKSIDDTSNFDDFPESDIL
QPVPNTTEPDYKSKDWVFLNYTYKRFEGLTQRGSIPTYMKAGKL
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM60589
n/a
NameBDBM60589
Synonyms:6-{[6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline (4) | BDBM50355498
Typen/a
Emp. Form.C18H13N7S
Mol. Mass.359.408
SMILESCn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1
Structure
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