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TargetCalcitonin gene-related peptide (CGRP alpha)
LigandBDBM50356279
Substrate/Competitorn/a
Meas. Tech.ChEMBL_775006
Ki 9.3±n/a nM
Citation Zartman CBBell IMGallicchio SNGraham SLKane SAMallee JJRutledge RZSalvatore CAVacca JPWilliams TM Identification of a novel RAMP-independent CGRP receptor antagonist. Bioorg Med Chem Lett 21:6705-8 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Calcitonin gene-related peptide (CGRP alpha)
Name:Calcitonin gene-related peptide (CGRP alpha)
Synonyms:CGRP | Calcitonin gene-related peptide 1
Type:Enzyme
Mol. Mass.:13902.80
Organism:Homo sapiens (Human)
Description:P06881
Residue:128
Sequence:
MGFQKFSPFLALSILVLLQAGSLHAAPFRSALESSPADPATLSEDEARLLLAALVQNYVQ
MKASELEQEQEREGSRIIAQKRACDTATCVTHRLAGLLSRSGGVVKNNFVPTNVGSKAFG
RRRRDLQA
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BDBM50356279
n/a
NameBDBM50356279
Synonyms:CHEMBL1910937
TypeSmall organic molecule
Emp. Form.C25H29Br2N5O4
Mol. Mass.623.337
SMILESCN(C)C(=O)[C@@H](Cc1cc(Br)c(O)c(Br)c1)NC(=O)N1CCC(CC1)N1Cc2ccccc2NC1=O |r|
Structure
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