Ki Summary

Reaction Details

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Target

Bcl-2-like protein 1

Ligand

BDBM50357759

Substrate/Competitor

n/a

Meas. Tech.

ChEMBL_785940 (CHEMBL1921340)

7.8±n/a nM

Citation

Goreshnik, I; Brock, AM; Maly, DJ Biochemical and pharmacological profiling of the pro-survival protein Bcl-xL. Bioorg Med Chem Lett21:4951-5 (2011) [PubMed] Article

More Info.:

Get all data from this article, Assay Method

Bcl-2-like protein 1

Name:

Bcl-2-like protein 1

Synonyms:

Type:

Mitochondrion membrane; Single-pass membrane protein

Mol. Mass.:

26039.60

Organism:

Homo sapiens (Human)

Description:

n/a

Residue:

233

Sequence:

MSQSNRELVVDFLSYKLSQKGYSWSQFSDVEENRTEAPEGTESEMETPSAINGNPSWHLA
DSPAVNGATGHSSSLDAREVIPMAAVKQALREAGDEFELRYRRAFSDLTSQLHITPGTAY
QSFEQVVNELFRDGVNWGRIVAFFSFGGALCVESVDKEMQVLVSRIAAWMATYLNDHLEP
WIQENGGWDTFVELYGNNAAAESRKGQERFNRWFLTGMTVAGVVLLGSLFSRK

BDBM50357759

n/a

Name

BDBM50357759

Synonyms:

CHEMBL1916197

Type

Small organic molecule

Emp. Form.

C108H170N32O31S

Mol. Mass.

2444.766

SMILES

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Structure