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TargetCasein kinase II subunit alpha'
LigandBDBM34038
Substrate/Competitorn/a
Meas. Tech.ChEMBL_792165 (CHEMBL1930612)
Ki 21±n/a nM
Citation Janeczko, MOrzeszko, AKazimierczuk, ZSzyszka, RBaier, A CK2a and CK2a' subunits differ in their sensitivity to 4,5,6,7-tetrabromo- and 4,5,6,7-tetraiodo-1H-benzimidazole derivatives. Eur J Med Chem47:345-50 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Casein kinase II subunit alpha'
Name:Casein kinase II subunit alpha'
Synonyms:CK2A2 | CSK22_HUMAN | CSNK2A2 | Casein kinase II alpha (prime) | Casein kinase II alpha' | Casein kinase II subunit alpha (CK2A2) | Casein kinase II subunit alpha (CSNK2A2)
Type:Protein
Mol. Mass.:41223.82
Organism:Homo sapiens (Human)
Description:n/a
Residue:350
Sequence:
MPGPAAGSRARVYAEVNSLRSREYWDYEAHVPSWGNQDDYQLVRKLGRGKYSEVFEAINI
TNNERVVVKILKPVKKKKIKREVKILENLRGGTNIIKLIDTVKDPVSKTPALVFEYINNT
DFKQLYQILTDFDIRFYMYELLKALDYCHSKGIMHRDVKPHNVMIDHQQKKLRLIDWGLA
EFYHPAQEYNVRVASRYFKGPELLVDYQMYDYSLDMWSLGCMLASMIFRREPFFHGQDNY
DQLVRIAKVLGTEELYGYLKKYHIDLDPHFNDILGQHSRKRWENFIHSENRHLVSPEALD
LLDKLLRYDHQQRLTAKEAMEHPYFYPVVKEQSQPCADNAVLSSGLTAAR
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  Blast E-value cutoff:
BDBM34038
n/a
NameBDBM34038
Synonyms:4,5,6,7-tetraiodobenzimidazole (TIBI), 1a
TypeSmall organic molecule
Emp. Form.C7H2I4N2
Mol. Mass.621.7221
SMILESIc1c(I)c(I)c2[nH]cnc2c1I
Structure
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