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TargetPeroxisome proliferator-activated receptor delta
LigandBDBM50360740
Substrate/Competitorn/a
Meas. Tech.ChEMBL_796446
EC50 2700±n/a nM
Citation Nomura MYumoto KShinozaki TIsogai STakano YMurakami K Discovery of cyclic amine-substituted benzoic acids as PPARa agonists. Bioorg Med Chem Lett 22:334-8 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Peroxisome proliferator-activated receptor delta
Name:Peroxisome proliferator-activated receptor delta
Synonyms:Nuclear receptor subfamily 1 group C member 2 | PPAR-beta | PPAR-delta | Peroxisome proliferator-activated receptor beta
Type:PROTEIN
Mol. Mass.:49786.42
Organism:Canis familiaris
Description:ChEMBL_796446
Residue:441
Sequence:
MEQPPGEAAEVREEEEKKEVAEAEGAPELNGGPERSLPSSSYTDLSRSSSPPSLLDQLQM
GGDGASCGSLNMECRVCGDKASGFHYGVHACEGCKGFFRRTIRMKLEYEKCERICKIQKK
NRNKCQYCRFQKCVALGMSHNAIRFGRMPEAEKRKLVAGLTANEGTQHNPQVADLKAFSK
HIYNAYLKNFNMTKKKARGILTGKASHTAPFVIHDIETLWQAEKGLVWKQLVNGLPPYKE
ISVHVFYRCQCTTVETVRELTEFAKSIPSFSNLFLNDQVTLLKYGVHEAIFAMLASIVNK
DGLLVANGTGFVTREFLRSLRKPFSDIIEPKFEFAVKFNALELDDSDLALFIAAIILCGD
RPGLINVPQVEAIQDTILRALEFHLQANHPYAQYLFPKLLQKMADLRQLVTEHAQMMQRI
KKTETETSLHPLLQEIYKDMY
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  Blast E-value cutoff:
BDBM50360740
n/a
NameBDBM50360740
Synonyms:CHEMBL1934476
TypeSmall organic molecule
Emp. Form.C23H22ClN3O3S
Mol. Mass.455.957
SMILESCc1nc(sc1C(=O)N[C@H]1CCCN(C1)c1cccc(c1)C(O)=O)-c1ccc(Cl)cc1 |r|
Structure
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