| Reaction Details |
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 | Report a problem with these data |
| Target | Glutathione S-transferase A2 |
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| Ligand | BDBM50361803 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_799590 (CHEMBL1941296) |
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| IC50 | >100000±n/a nM |
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| Citation |  Wang, CH; Wu, HT; Cheng, HM; Yen, TJ; Lu, IH; Chang, HC; Jao, SC; Shing, TK; Li, WS Inhibition of glutathione S-transferase M1 by new gabosine analogues is essential for overcoming cisplatin resistance in lung cancer cells. J Med Chem54:8574-81 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| |
| Glutathione S-transferase A2 |
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| Name: | Glutathione S-transferase A2 |
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| Synonyms: | GST class-alpha member 2 | GST-gamma | GST2 | GSTA2 | GSTA2-2 | GSTA2_HUMAN | GTH2 | HA subunit 2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 25667.17 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_799590 |
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| Residue: | 222 |
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| Sequence: | MAEKPKLHYSNIRGRMESIRWLLAAAGVEFEEKFIKSAEDLDKLRNDGYLMFQQVPMVEI
DGMKLVQTRAILNYIASKYNLYGKDIKEKALIDMYIEGIADLGEMILLLPFSQPEEQDAK
LALIQEKTKNRYFPAFEKVLKSHGQDYLVGNKLSRADIHLVELLYYVEELDSSLISSFPL
LKALKTRISNLPTVKKFLQPGSPRKPPMDEKSLEESRKIFRF
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| BDBM50361803 |
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| n/a |
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| Name | BDBM50361803 |
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| Synonyms: | CHEMBL1938620 |
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| Type | Small organic molecule |
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| Emp. Form. | C9H12O6 |
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| Mol. Mass. | 216.188 |
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| SMILES | CC(=O)OCC1C[C@H](O)[C@H](O)C(=O)C1=O |r| |
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| Structure | 
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