| Reaction Details |
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 | Report a problem with these data |
| Target | Prostaglandin D2 receptor 2 |
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| Ligand | BDBM50362158 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_797760 (CHEMBL1944119) |
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| IC50 | >1000±n/a nM |
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| Citation |  Ito, S; Terasaka, T; Zenkoh, T; Matsuda, H; Hayashida, H; Nagata, H; Imamura, Y; Kobayashi, M; Takeuchi, M; Ohta, M Discovery of novel and potent CRTH2 antagonists. Bioorg Med Chem Lett22:1194-7 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Prostaglandin D2 receptor 2 |
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| Name: | Prostaglandin D2 receptor 2 |
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| Synonyms: | Chemoattractant receptor-homologous molecule expressed on Th2 cells |
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| Type: | PROTEIN |
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| Mol. Mass.: | 42241.65 |
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| Organism: | Cavia porcellus |
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| Description: | ChEMBL_797760 |
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| Residue: | 391 |
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| Sequence: | MANATLKPLCPVLKDMSLLGSHSNSSLRYMDHISVLLHGLAALLGLVENGLIVFVVGCRM
RQTVVTTWALHLALSDLLASAALPFFTYFLAVGHSWELGTAFCKLHSSVFFLNMFASGFL
LSAISLDRCVRVVHPVWAQNHRSVSVARRVCAVLWALALLNTVPYFVFRDTILRRDGRTM
CYYNVLLLAPAGDHNATCGTRQMALALSKFLLAFALPLGIIAASHAVVSARLQRRPQGGV
RPGRFVRLVAAVVAAFALCWGPYHAFSLIEARAHAVPSLRPLAWRALPFVSSLAFINSVV
NPLLYVLTCPDVGRKLRRSLRAVLESVLVDDGELGSRYRRRGGSSSPAVASASSSLSLAP
ATHQACSLLRWLRGSRGTGSDDAPSSASGQG
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| BDBM50362158 |
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| n/a |
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| Name | BDBM50362158 |
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| Synonyms: | CHEMBL1941119 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H25Cl2NO4 |
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| Mol. Mass. | 522.419 |
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| SMILES | OC(=O)COc1cccc(CCCn2cc(ccc2=O)C(c2ccc(Cl)cc2)c2ccc(Cl)cc2)c1 |
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| Structure | 
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