| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50365855 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_806706 (CHEMBL1958666) |
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| Ki | 0.1±n/a nM |
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| Citation |  Lunn, G; Roberts, LR; Content, S; Critcher, DJ; Douglas, S; Fenwick, AE; Gethin, DM; Goodwin, G; Greenway, D; Greenwood, S; Hall, K; Thomas, M; Thompson, S; Williams, D; Wood, G; Wylie, A SAR and biological evaluation of 3-azabicyclo[3.1.0]hexane derivatives asµ opioid ligands. Bioorg Med Chem Lett22:2200-3 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1 |
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| Type: | G Protein-Coupled Receptor (GPCR) |
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| Mol. Mass.: | 44789.51 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P35372 |
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| Residue: | 400 |
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| Sequence: | MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCP
PTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALAT
STLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDF
RTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFI
FAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHI
YVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNI
EQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP
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| BDBM50365855 |
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| n/a |
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| Name | BDBM50365855 |
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| Synonyms: | CHEMBL1957843 |
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| Type | Small organic molecule |
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| Emp. Form. | C24H30N2O3S |
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| Mol. Mass. | 426.572 |
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| SMILES | CC[C@]1([C@H]2CN(CC3Cc4ccccc4C3O)C[C@@H]12)c1cccc(NS(C)(=O)=O)c1 |r| |
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| Structure | 
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