| Reaction Details |
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 | Report a problem with these data |
| Target | Platelet-activating factor receptor |
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| Ligand | BDBM50366241 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_155156 (CHEMBL760196) |
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| Ki | 103±n/a nM |
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| Citation |  Sahoo, SP; Graham, DW; Acton, J; Biftu, T; Bugianesi, RL; Girotra, NN; Kuo, C; Ponpipom, MM; Doebber, TW; Wu, MS; Hwang, S; Lam, M; MacIntyre, D; Bach, TJ; Luell, S; Meurer, R; Davies, P; Alberts, AW; Chabala, JC Synthesis and biological activity of MK 287 (L-680,573): a potent, specific and orally active paf receptor antagonist Bioorg Med Chem Lett1:327-332 (1991) Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Platelet-activating factor receptor |
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| Name: | Platelet-activating factor receptor |
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| Synonyms: | PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor |
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| Type: | Protein |
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| Mol. Mass.: | 39005.63 |
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| Organism: | Cavia porcellus |
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| Description: | n/a |
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| Residue: | 342 |
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| Sequence: | MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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| BDBM50366241 |
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| n/a |
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| Name | BDBM50366241 |
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| Synonyms: | CHEMBL297624 | L-652731 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H28O7 |
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| Mol. Mass. | 404.4535 |
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| SMILES | COc1cc(cc(OC)c1OC)[C@H]1CC[C@@H](O1)c1cc(OC)c(OC)c(OC)c1 |
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| Structure | 
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