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Reaction Details
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TargetPhospholipase A2
LigandBDBM50015214
Substrate/Competitorn/a
Meas. Tech.ChEBML_156506
IC50 100000±n/a nM
Citation Wilkerson, WDeLucca, IGalbraith, WHarris, RKerr, J Antiinflammatory -benzeneethanamines. III Bioorg Med Chem Lett3:711-716 (1993)    Article
More Info.:Get all data from this article,  Assay Method
 
Phospholipase A2
Name:Phospholipase A2
Synonyms:PA21B_RAT | Phospholipase A2 group 1B | Pla2g1b
Type:PROTEIN
Mol. Mass.:16427.59
Organism:Rattus norvegicus
Description:ChEMBL_156506
Residue:146
Sequence:
MKLLLLAALLTAGVTAHSISTRAVWQFRNMIKCTIPGSDPLREYNNYGCYCGLGGSGTPV
DDLDRCCQTHDHCYNQAKKLESCKFLIDNPYTNTYSYKCSGNVITCSDKNNDCESFICNC
DRQAAICFSKVPYNKEYKDLDTKKHC
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  Blast E-value cutoff:
BDBM50015214
n/a
NameBDBM50015214
Synonyms:6-chloro-2-methoxy-9-acridinyl(4-diethylamino-1-methylbutyl)amine | 6-chloro-N-(5-(diethylamino)pentan-2-yl)-2-methoxyacridin-9-amine | CHEMBL7568 | N'-(6-chloro-2-methoxy-acridin-9-yl)-N,N-diethyl-pentane-1,4-diamine | N*4*-(6-Chloro-2-methoxy-acridin-9-yl)-N*1*,N*1*-diethyl-pentane-1,4-diamine | N*4*-(6-Chloro-2-methoxy-acridin-9-yl)-N*1*,N*1*-diethyl-pentane-1,4-diamine (Mepacrine) | N*4*-(6-Chloro-2-methoxy-acridin-9-yl)-N*1*,N*1*-diethyl-pentane-1,4-diamine ; (mepacrine) | N-(4-Hydroxy-phenyl)-acetamide | cid_237 | quinacrine
TypeSmall organic molecule
Emp. Form.C23H30ClN3O
Mol. Mass.399.957
SMILESCCN(CC)CCCC(C)Nc1c2ccc(Cl)cc2nc2ccc(OC)cc12
Structure
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