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TargetRetinoid receptor
LigandBDBM50290079
Substrate/Competitorn/a
Meas. Tech.ChEBML_195497
Ki 90±n/a nM
Citation Diaz PMichel SStella LCharpentier B Synthesis and biological activities of new heterocyclic aromatic retinoids Bioorg Med Chem Lett 7:2289-2294 (1997)    Article
More Info.:Get all data from this article,  Assay Method
 
Retinoid receptor
Name:Retinoic acid receptor RXR-alpha/Retinoic acid receptor beta
Synonyms:HBV-activated protein | Nuclear receptor subfamily 1 group B member 2 | RAR-beta | RAR-epsilon | Retinoic acid receptor beta
Type:PROTEIN
Mol. Mass.:50498.70
Organism:Homo sapiens (Human)
Description:ChEMBL_1458015
Residue:455
Sequence:
MTTSGHACPVPAVNGHMTHYPATPYPLLFPPVIGGLSLPPLHGLHGHPPPSGCSTPSPAT
IETQSTSSEELVPSPPSPLPPPRVYKPCFVCQDKSSGYHYGVSACEGCKGFFRRSIQKNM
IYTCHRDKNCVINKVTRNRCQYCRLQKCFEVGMSKESVRNDRNKKKKETSKQECTESYEM
TAELDDLTEKIRKAHQETFPSLCQLGKYTTNSSADHRVRLDLGLWDKFSELATKCIIKIV
EFAKRLPGFTGLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNA
GFGPLTDLVFTFANQLLPLEMDDTETGLLSAICLICGDRQDLEEPTKVDKLQEPLLEALK
IYIRKRRPSKPHMFPKILMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLENSEGH
EPLTPSSSGNTAEHSPSISPSSVENSGVSQSPLVQ
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  Blast E-value cutoff:
BDBM50290079
n/a
NameBDBM50290079
Synonyms:3-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthalen-2-yl)-chroman-7-carboxylic acid | CHEMBL75527
TypeSmall organic molecule
Emp. Form.C24H28O3
Mol. Mass.364.4773
SMILESCC1(C)CCC(C)(C)c2cc(ccc12)C1COc2cc(ccc2C1)C(O)=O
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: