| Reaction Details |
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 | Report a problem with these data |
| Target | Muscarinic acetylcholine receptor M5 |
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| Ligand | BDBM81462 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEBML_139800 |
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| IC50 | 10±n/a nM |
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| Citation |  Augelli-Szafran, CE; Jaen, JC; Moreland, DW; Nelson, CB; Penvose-Yi, JR; Schwarz, RD Identification and characterization of m4 selective muscarinic antagonists. Bioorg Med Chem Lett8:1991-6 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Muscarinic acetylcholine receptor M5 |
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| Name: | Muscarinic acetylcholine receptor M5 |
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| Synonyms: | ACM5_HUMAN | CHRM5 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 60102.35 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1517990 |
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| Residue: | 532 |
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| Sequence: | MEGDSYHNATTVNGTPVNHQPLERHRLWEVITIAAVTAVVSLITIVGNVLVMISFKVNSQ
LKTVNNYYLLSLACADLIIGIFSMNLYTTYILMGRWALGSLACDLWLALDYVASNASVMN
LLVISFDRYFSITRPLTYRAKRTPKRAGIMIGLAWLISFILWAPAILCWQYLVGKRTVPL
DECQIQFLSEPTITFGTAIAAFYIPVSVMTILYCRIYRETEKRTKDLADLQGSDSVTKAE
KRKPAHRALFRSCLRCPRPTLAQRERNQASWSSSRRSTSTTGKPSQATGPSANWAKAEQL
TTCSSYPSSEDEDKPATDPVLQVVYKSQGKESPGEEFSAEETEETFVKAETEKSDYDTPN
YLLSPAAAHRPKSQKCVAYKFRLVVKADGNQETNNGCHKVKIMPCPFPVAKEPSTKGLNP
NPSHQMTKRKRVVLVKERKAAQTLSAILLAFIITWTPYNIMVLVSTFCDKCVPVTLWHLG
YWLCYVNSTVNPICYALCNRTFRKTFKMLLLCRWKKKKVEEKLYWQGNSKLP
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| BDBM81462 |
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| n/a |
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| Name | BDBM81462 |
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| Synonyms: | (R)-Trihexyphenidyl | (S)-Trihexyphenidyl | Benzhexol | CAS_58947-95-8 | NSC_5572 | TRIHEXYPHENIDYL HYDROCHLORIDE | Trihexyphenidyl |
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| Type | Small organic molecule |
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| Emp. Form. | C20H31NO |
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| Mol. Mass. | 301.4662 |
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| SMILES | OC(CCN1CCCCC1)(C1CCCCC1)c1ccccc1 |
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| Structure | 
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