| Reaction Details |
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 | Report a problem with these data |
| Target | Glutamyl aminopeptidase |
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| Ligand | BDBM50078120 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_32826 (CHEMBL646477) |
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| Ki | 0.000±n/a nM |
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| Comments | Zero 01/04/22 |
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| Citation |  Chen, H; Roques, BP; Fournié-Zaluski, MC Design of the first highly potent and selective aminopeptidase N (EC 3.4.11.2) inhibitor. Bioorg Med Chem Lett9:1511-6 (1999) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Glutamyl aminopeptidase |
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| Name: | Glutamyl aminopeptidase |
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| Synonyms: | AMPE_PIG | APA | Aminopeptidase A | CD_antigen=CD249 | EAP | ENPEP | Glutamyl aminopeptidase |
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| Type: | PROTEIN |
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| Mol. Mass.: | 108259.08 |
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| Organism: | Sus scrofa |
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| Description: | ChEMBL_32826 |
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| Residue: | 942 |
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| Sequence: | MSTDSKRYCIKTKHVAIICAAVVAVGLIVGLSVGLTRSCDSKDGGQGTTQSPSHLPPTSS
PPQDQGVCPASEDESGNWRDFRLPDFINPVHYDLQVKPLLEQDTYTGTVNISINVTSPTQ
HLWLHLRETRITQLPVLWRPSGEQVQVRRCFEYKKQEYVVVEAEEELAPNSGEGLYHLTM
EFAGWLNGSLVGFYRTTYVEKGQIKSIAATDHEPTDARKSFPCFDEPNKKATYTISIIHP
KEYKALSNMPVEKEESVDDIWTQTTFQKSVPMSTYLVCFAVHQFDSVTRTSRSGKPLTIY
VQPEQKHTAEYAANITKSVFDYFEDYFAMEYSLPKLDKIAIPDFGTGAMENWGLITYRET
NLLYDPNESASSNQQRVAAVVAHELVHQWFGNIVTMEWWEDLWLNEGFASFFEFLGVDHA
EKEWQMRDQILLEDVLPVQEDDSLISSHPIVVTVSTPAEITSVFDGISYSKGASILRMLE
DWITPEKFQKGCQEYLKKFEFKNAKTSDFWEALEEASNLPVKEVMDTWTNQMGYPVLNVE
DMRIISQKRFLLDPNANSSEPHSVFGYTWNIPVRWTNDNESTITIYNRSETGGITLNSSN
PNGNAFLKINPDHIGFYRVNYEVSTWEWIATNLSLNHKDFSTADRASLIDDAFALARAQL
LNYKEALNLTKYLKMEDEYLPWQRVISAVTYIISMFEDDKELYPMIEKYFRDQVKPIADS
LGWNDNGDHLTKLLRASVLGFACKMGDSNALNNASHLFEQWLTGTVSLPVNLRLLVYRYG
MQNSGNETSWNYTLKQYQETSLAQEKEKLLYGLASVKNVALLSRYLDLLKDPNVIKSQDV
FTVIRYISYNSYGKTMAWNWIQLNWEYLVNRYTLNDRNLGRIVTIAEPFNTELQLWQMES
FFKRYPEAGAGEKPREQVLETVKNNIEWLKQNRDTIRDWFFN
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| BDBM50078120 |
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| n/a |
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| Name | BDBM50078120 |
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| Synonyms: | (R)-1-{[(S)-2-((S)-1-Carboxy-1-methyl-2-phenyl-ethylcarbamoyl)-3-phenyl-propyl]-hydroxy-phosphinoyl}-ethyl-ammonium |
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| Type | Small organic molecule |
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| Emp. Form. | C22H30N2O5P |
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| Mol. Mass. | 433.4572 |
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| SMILES | C[C@H]([NH3+])P(O)(=O)C[C@@H](Cc1ccccc1)C(=O)N[C@@](C)(Cc1ccccc1)C(O)=O |
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| Structure | 
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