Ki Summary BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetMu-type opioid receptor
LigandBDBM50369586
Substrate/Competitorn/a
Meas. Tech.ChEMBL_145278 (CHEMBL751214)
Ki 1.1±n/a nM
Citation Wentland, MPXu, GCioffi, CLYe, YDuan, WCohen, DJColasurdo, AMBidlack, JM 8-Aminocyclazocine analogues: synthesis and structure-activity relationships. Bioorg Med Chem Lett10:183-7 (2000) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50369586
n/a
NameBDBM50369586
Synonyms:CHEMBL326516
TypeSmall organic molecule
Emp. Form.C24H30N2
Mol. Mass.346.5084
SMILESC[C@H]1[C@H]2Cc3ccc(Nc4ccccc4)cc3[C@@]1(C)CCN2CC1CC1 |TLB:22:21:1:16.4.3|
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: