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TargetMu-type opioid receptor
LigandBDBM50017233
Substrate/Competitorn/a
Meas. Tech.ChEBML_145282
Ki 0.210000±n/a nM
Citation Neumeyer JLGu XHvan Vliet LADeNunzio NJRusovici DECohen DJNegus SSMello NKBidlack JM Mixed kappa agonists and mu agonists/antagonists as potential pharmacotherapeutics for cocaine abuse: synthesis and opioid receptor binding affinity of N-substituted derivatives of morphinan. Bioorg Med Chem Lett 11:2735-40 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50017233
n/a
NameBDBM50017233
Synonyms:CHEMBL592 | LEVO-DROMORAN | LEVORPHANOL
TypeSmall organic molecule
Emp. Form.C17H23NO
Mol. Mass.257.3706
SMILESCN1CC[C@]23CCCC[C@H]2[C@H]1Cc1ccc(O)cc31 |r,TLB:0:1:12.18.11:9|
Structure
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