| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 3 |
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| Ligand | BDBM50219321 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_200508 (CHEMBL803852) |
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| Ki | 1200±n/a nM |
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| Citation |  Contour-Galéra, MO; Poitout, L; Moinet, C; Morgan, B; Gordon, T; Roubert, P; Thurieau, C Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5. Bioorg Med Chem Lett11:741-5 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 3 |
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| Name: | Somatostatin receptor type 3 |
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| Synonyms: | SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3) |
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| Type: | Protein |
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| Mol. Mass.: | 45855.97 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P32745 |
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| Residue: | 418 |
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| Sequence: | MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLL
GNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVM
AVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVV
FSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRV
WAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVA
LPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEE
SREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
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| BDBM50219321 |
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| n/a |
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| Name | BDBM50219321 |
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| Synonyms: | CHEMBL2112934 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H34N6O |
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| Mol. Mass. | 494.6306 |
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| SMILES | CC(C)(C(=O)NCCc1c[nH]c2ccccc12)c1cn2cc(Cc3ccccc3)nc(CCCN)c2n1 |
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| Structure | 
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