| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 1 |
|---|
| Ligand | BDBM50099176 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_225192 |
|---|
| Ki | 2570±n/a nM |
|---|
| Citation |  Moinet, C; Contour-Galcéra, MO; Poitout, L; Morgan, B; Gordon, T; Rouber, P; Thurieau, C Novel non-peptide ligands for the somatostatin sst3 receptor. Bioorg Med Chem Lett11:991-5 (2001) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 1 |
|---|
| Name: | Somatostatin receptor type 1 |
|---|
| Synonyms: | SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 42692.81 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P30872 |
|---|
| Residue: | 391 |
|---|
| Sequence: | MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAIL
ISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLL
RHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLG
VWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAIC
LCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQD
DATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKS
RAYSVEDFQPENLESGGVFRNGTCTSRITTL
|
|
|
|---|
| BDBM50099176 |
|---|
| n/a |
|---|
| Name | BDBM50099176 |
|---|
| Synonyms: | CHEMBL176313 | N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-4-trifluoromethoxy-benzamidine |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C27H22F3N5O |
|---|
| Mol. Mass. | 489.4917 |
|---|
| SMILES | NC(=N[C@H](Cc1c[nH]c2ccccc12)c1nc(c[nH]1)-c1ccccc1)c1ccc(OC(F)(F)F)cc1 |w:1.0| |
|---|
| Structure | 
|
|---|
Search and Browse
