| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Beta-galactoside alpha-2,6-sialyltransferase 1 |
|---|
| Ligand | BDBM50366833 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_216152 (CHEMBL817949) |
|---|
| Ki | 730000±n/a nM |
|---|
| Citation |  Whalen, LJ; McEvoy, KA; Halcomb, RL Synthesis and evaluation of phosphoramidate amino acid-based inhibitors of sialyltransferases. Bioorg Med Chem Lett13:301-4 (2002) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Beta-galactoside alpha-2,6-sialyltransferase 1 |
|---|
| Name: | Beta-galactoside alpha-2,6-sialyltransferase 1 |
|---|
| Synonyms: | CMP-N-acetylneuraminate-beta-galactosamide-alpha-2,6-sialyltransferase | SIAT1_RAT | Siat1 | St6gal1 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 46743.36 |
|---|
| Organism: | Rattus norvegicus |
|---|
| Description: | ChEMBL_216152 |
|---|
| Residue: | 403 |
|---|
| Sequence: | MIHTNLKKKFSLFILVFLLFAVICVWKKGSDYEALTLQAKEFQMPKSQEKVAMGSASQVV
FSNSKQDPKEDIPILSYHRVTAKVKPQPSFQVWDKDSTYSKLNPRLLKIWRNYLNMNKYK
VSYKGPGPGVKFSVEALRCHLRDHVNVSMIEATDFPFNTTEWEGYLPKENFRTKVGPWQR
CAVVSSAGSLKNSQLGREIDNHDAVLRFNGAPTDNFQQDVGSKTTIRLMNSQLVTTEKRF
LKDSLYTEGILIVWDPSVYHADIPKWYQKPDYNFFETYKSYRRLNPSQPFYILKPQMPWE
LWDIIQEISADLIQPNPPSSGMLGIIIMMTLCDQVDIYEFLPSKRKTDVCYYHQKFFDSA
CTMGAYDPLLFEKNMVKHLNEGTDEDIYLFGKATLSGFRNIRC
|
|
|
|---|
| BDBM50366833 |
|---|
| n/a |
|---|
| Name | BDBM50366833 |
|---|
| Synonyms: | CHEMBL608928 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H24N5O9P |
|---|
| Mol. Mass. | 509.4064 |
|---|
| SMILES | Nc1ccn(C2O[C@H](COP(O)(=O)N[C@@H](Cc3c[nH]c4ccccc34)C(O)=O)[C@@H](O)[C@H]2O)c(=O)n1 |r| |
|---|
| Structure | 
|
|---|
Search and Browse
