| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Adenosine receptor A3 |
|---|
| Ligand | BDBM50366923 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_31701 |
|---|
| Ki | >10000±n/a nM |
|---|
| Citation |  Dukat, M; Taroua, M; Dahdouh, A; Siripurapu, U; Damaj, MI; Martin, BR; Glennon, RA (+/-)8-Amino-5,6,7,8-tetrahydroisoquinolines as novel antinociceptive agents. Bioorg Med Chem Lett14:3651-4 (2004) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Adenosine receptor A3 |
|---|
| Name: | Adenosine receptor A3 |
|---|
| Synonyms: | A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR) |
|---|
| Type: | G Protein-Coupled Receptor (GPCR) |
|---|
| Mol. Mass.: | 36197.32 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P0DMS8 |
|---|
| Residue: | 318 |
|---|
| Sequence: | MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIA
VGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKR
VTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYF
SFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFA
LSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKAC
VVCHPSDSLDTSIEKNSE
|
|
|
|---|
| BDBM50366923 |
|---|
| n/a |
|---|
| Name | BDBM50366923 |
|---|
| Synonyms: | CHEMBL1794855 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C12H18N2 |
|---|
| Mol. Mass. | 190.2847 |
|---|
| SMILES | CCN(C)C1CCCc2ccncc12 |
|---|
| Structure | 
|
|---|
Search and Browse
