Reaction Details | |||
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Target | Transporter | ||
Ligand | BDBM50005548 | ||
Substrate/Competitor | n/a | ||
Meas. Tech. | ChEBML_144836 | ||
IC50 | 6.6±n/a nM | ||
Citation | Bøgesø, KP Neuroleptic activity and dopamine-uptake inhibition in 1-piperazino-3-phenylindans. J Med Chem26:935-47 (1983) [PubMed] | ||
More Info.: | Get all data from this article, Assay Method | ||
Transporter | |||
Name: | Transporter | ||
Synonyms: | Monoamine transporters; Norepininephrine & dopamine | Norepinephrine Monoamine transporters | ||
Type: | PROTEIN | ||
Mol. Mass.: | 66787.87 | ||
Organism: | Rattus norvegicus | ||
Description: | ChEMBL_1463061 | ||
Residue: | 597 | ||
Sequence: |
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BDBM50005548 | |||
n/a | |||
Name | BDBM50005548 | ||
Synonyms: | (+)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | (+/-)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | (-)-2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | (Nomifensine) 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine (Nomifensine) | 2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine(Nomifensine) | 2-methyl-4-phenyl-1,2,3,4-tetrahydroisoquinolin-8-amine | CHEMBL273575 | NOMIFENSINE | NOMIFENSINE2-Methyl-4-phenyl-1,2,3,4-tetrahydro-isoquinolin-8-ylamine | ||
Type | Small organic molecule | ||
Emp. Form. | C16H18N2 | ||
Mol. Mass. | 238.3275 | ||
SMILES | CN1CC(c2ccccc2)c2cccc(N)c2C1 | ||
Structure |