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TargetThymidine kinase, cytosolic
LigandBDBM50207303
Substrate/Competitorn/a
Meas. Tech.ChEBML_208005
Ki 5060±n/a nM
Citation Efange SMAlessi EMShih HCCheng YCBardos TJ Synthesis and biological activities of 2-pyrimidinone nucleosides. 2. 5-Halo-2-pyrimidinone 2'-deoxyribonucleosides. J Med Chem 28:904-10 (1985) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Thymidine kinase, cytosolic
Name:Thymidine kinase, cytosolic
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:25476.50
Organism:Homo sapiens (Human)
Description:ChEMBL_1333884
Residue:234
Sequence:
MSCINLPTVLPGSPSKTRGQIQVILGPMFSGKSTELMRRVRRFQIAQYKCLVIKYAKDTR
YSSSFCTHDRNTMEALPACLLRDVAQEALGVAVIGIDEGQFFPDIVEFCEAMANAGKTVI
VAALDGTFQRKPFGAILNLVPLAESVVKLTAVCMECFREAAYTKRLGTEKEVEVIGGADK
YHSVCRLCYFKKASGQPAGPDNKENCPVPGKPGEAVAARKLFAPQQILQCSPAN
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BDBM50207303
n/a
NameBDBM50207303
Synonyms:5-BROMO-2'-DEOXY URIDINE | 5-bromo-1-((2R,4S,5R)-4-hydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)pyrimidine-2,4(1H,3H)-dione | Bromodeoxyuridine | CHEMBL222280 | cid_6035
TypeSmall organic molecule
Emp. Form.C9H11BrN2O5
Mol. Mass.307.098
SMILESOC[C@H]1O[C@H](C[C@@H]1O)n1cc(Br)c(=O)[nH]c1=O |r|
Structure
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