| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Muscarinic receptor M1 |
|---|
| Ligand | BDBM39341 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_140160 |
|---|
| Ki | 3.6±n/a nM |
|---|
| Citation |  Rzeszotarski, WJ; McPherson, DW; Ferkany, JW; Kinnier, WJ; Noronha-Blob, L; Kirkien-Rzeszotarski, A Affinity and selectivity of the optical isomers of 3-quinuclidinyl benzilate and related muscarinic antagonists. J Med Chem31:1463-6 (1988) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Muscarinic receptor M1 |
|---|
| Name: | Muscarinic receptor M1 |
|---|
| Synonyms: | Muscarinic acetylcholine receptor M1 |
|---|
| Type: | PROTEIN |
|---|
| Mol. Mass.: | 15022.43 |
|---|
| Organism: | Bos taurus |
|---|
| Description: | ChEMBL_140161 |
|---|
| Residue: | 139 |
|---|
| Sequence: | ETENRARELAALQGSETPGKGGGSSSSSERSQPGAEGSPETPPGRCCRCCRTPRLLQAYS
WKEEEEEDEGSMESLTSSEGEEPGSEVVIKMPMVDPEAQAPAKQPPRSSPNTVKRPTRKG
RERAGKGQKPRGKEQLAKR
|
|
|
|---|
| BDBM39341 |
|---|
| n/a |
|---|
| Name | BDBM39341 |
|---|
| Synonyms: | 11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one | 11-[2-(4-methyl-1-piperazinyl)-1-oxoethyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;hydrochloride | 11-[2-(4-methylpiperazin-1-yl)acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;hydrochloride | 11-[2-(4-methylpiperazin-1-yl)ethanoyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;hydrochloride | 11-[2-(4-methylpiperazino)acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;hydrochloride | CHEMBL9967 | MLS000069702 | PIRENZEPINE | PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | cid_185248 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H21N5O2 |
|---|
| Mol. Mass. | 351.4023 |
|---|
| SMILES | CN1CCN(CC(=O)N2c3ccccc3C(=O)Nc3cccnc23)CC1 |
|---|
| Structure | 
|
|---|
Search and Browse
