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TargetMuscarinic acetylcholine receptor M1
LigandBDBM50403547
Substrate/Competitorn/a
Meas. Tech.ChEBML_138126
Ki 2.4±n/a nM
Citation Leader HSmejkal RMPayne CSPadilla FNDoctor BPGordon RKChiang PK Binary antidotes for organophosphate poisoning: aprophen analogues that are both antimuscarinics and carbamates. J Med Chem 32:1522-8 (1989) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Muscarinic acetylcholine receptor M1
Name:Muscarinic acetylcholine receptor M1
Synonyms:n/a
Type:PROTEIN
Mol. Mass.:15022.43
Organism:Bos taurus
Description:ChEMBL_140161
Residue:139
Sequence:
ETENRARELAALQGSETPGKGGGSSSSSERSQPGAEGSPETPPGRCCRCCRTPRLLQAYS
WKEEEEEDEGSMESLTSSEGEEPGSEVVIKMPMVDPEAQAPAKQPPRSSPNTVKRPTRKG
RERAGKGQKPRGKEQLAKR
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  Blast E-value cutoff:
BDBM50403547
n/a
NameBDBM50403547
Synonyms:ATROPEN | ATROPINE
TypeSmall organic molecule
Emp. Form.C17H23NO3
Mol. Mass.289.3694
SMILESCN1[C@H]2CC[C@@H]1C[C@@H](C2)OC(=O)C(CO)c1ccccc1 |r,THB:9:7:1:3.4|
Structure
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