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TargetChymotrypsinogen A
LigandBDBM50014578
Substrate/Competitorn/a
Meas. Tech.ChEBML_216617
Ki 60±n/a nM
Citation Angelastro, MRMehdi, SBurkhart, JPPeet, NPBey, P Alpha-diketone and alpha-keto ester derivatives of N-protected amino acids and peptides as novel inhibitors of cysteine and serine proteinases. J Med Chem33:11-3 (1990) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Chymotrypsinogen A
Name:Chymotrypsinogen A
Synonyms:Alpha-chymotrypsin | CTRA_BOVIN | Chymotrypsin A | Chymotrypsin A chain A | Chymotrypsin A chain B | Chymotrypsin A chain C | Chymotrypsinogen A | alpha-Chymotrypsin (α-Chymotrypsin)
Type:Serine protease
Mol. Mass.:25670.88
Organism:Bos taurus (bovine)
Description:n/a
Residue:245
Sequence:
CGVPAIQPVLSGLSRIVNGEEAVPGSWPWQVSLQDKTGFHFCGGSLINENWVVTAAHCGV
TTSDVVVAGEFDQGSSSEKIQKLKIAKVFKNSKYNSLTINNDITLLKLSTAASFSQTVSA
VCLPSASDDFAAGTTCVTTGWGLTRYTNANTPDRLQQASLPLLSNTNCKKYWGTKIKDAM
ICAGASGVSSCMGDSGGPLVCKKNGAWTLVGIVSWGSSTCSTSTPGVYARVTALVNWVQQ
TLAAN
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  Blast E-value cutoff:
BDBM50014578
n/a
NameBDBM50014578
Synonyms:3-(2-Benzyloxycarbonylamino-3-methyl-butyrylamino)-2-oxo-4-phenyl-butyric acid methyl ester | CHEMBL282374
TypeSmall organic molecule
Emp. Form.C24H28N2O6
Mol. Mass.440.4889
SMILESCOC(=O)C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C
Structure
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