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TargetSex hormone-binding globulin
LigandBDBM50367916
Substrate/Competitorn/a
Meas. Tech.ChEBML_35818
IC50 3.7±n/a nM
Citation Winneker, RCWagner, MMSingh, B A novel, nonsteroidal inhibitor of androgen binding to the rat androgen binding protein: diethyl [[[3-(2,6-dimethyl-4-pyridinyl)-4-fluorophenyl]amino]methylene] propanedioate. J Med Chem33:129-32 (1990) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Sex hormone-binding globulin
Name:Sex hormone-binding globulin
Synonyms:ABP | SBP | SHBG_RAT | Sex hormone-binding globulin | Sex steroid-binding protein | Shbg | Testis-specific androgen-binding protein
Type:PROTEIN
Mol. Mass.:44530.46
Organism:Rattus norvegicus
Description:ChEMBL_35819
Residue:403
Sequence:
MEKGEVASLRCRLLLLLLLLTLPPTHQGRTLRHIDPIQSAQDSPAKYLSNGPGQEPVTVL
TIDLTKISKPSSSFEFRTWDPEGVIFYGDTNTEDDWFMLGLRDGQLEIQLHNLWARLTVG
FGPRLNDGRWHPVELKMNGDSLLLWVDGKEMLCLRQVSASLADHPQLSMRIALGGLLLPT
SKLRFPLVPALDGCIRRDIWLGHQAQLSTSARTSLGNCDVDLQPGLFFPPGTHAEFSLQD
IPQPHTDPWTFSLELGFKLVDGAGRLLTLGTGTNSSWLTLHLQDQTVVLSSEAEPKLALP
LAVGLPLQLKLDVFKVALSQGPKMEVLSTSLLRLASLWRLWSHPQGHLSLGALPGEDSSA
SFCLSDLWVQGQRLDIDKALSRSQDIWTHSCPQSPSNDTHTSH
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  Blast E-value cutoff:
BDBM50367916
n/a
NameBDBM50367916
Synonyms:METHYLTRIENOLONE | Metribolone | R-1881
TypeSmall organic molecule
Emp. Form.C19H24O2
Mol. Mass.284.3927
SMILESC[C@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CCC4=C3C=C[C@]12C |r,c:16,19,t:9|
Structure
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