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TargetPlatelet activating factor receptor
LigandBDBM50014004
Substrate/Competitorn/a
Meas. Tech.ChEBML_155157
Ki 1001±n/a nM
Citation Sunkel CEde Casa-Juana MFSantos LGómez MMVillarroya MGonzález-Morales MAPriego JGOrtega MP 4-Alkyl-1,4-dihydropyridines derivatives as specific PAF-acether antagonists. J Med Chem 33:3205-10 (1991) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Platelet activating factor receptor
Name:Platelet activating factor receptor
Synonyms:PAF-R | Platelet-activating factor receptor
Type:Protein
Mol. Mass.:39005.63
Organism:Cavia porcellus
Description:n/a
Residue:342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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  Blast E-value cutoff:
BDBM50014004
n/a
NameBDBM50014004
Synonyms:2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxylic acid 3-ethyl ester 5-(2-ethylsulfanyl-ethyl) ester | CHEMBL108714
TypeSmall organic molecule
Emp. Form.C16H25NO4S
Mol. Mass.327.439
SMILESCCOC(=O)C1C(C)C(C(=O)OCCSCC)=C(C)N=C1C |c:19,t:16|
Structure
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